The third transmembrane helix of the cannabinoid receptor plays a role in the selectivity of aminoalkylindoles for CB2, peripheral cannabinoid receptor. [electronic resource]
Producer: 19991124Description: 837-44 p. digitalISSN:- 0022-3565
- Animals
- Benzoxazines
- Binding Sites
- CHO Cells -- physiology
- Central Nervous System -- physiology
- Cloning, Organism
- Colforsin -- pharmacology
- Cricetinae
- Cyclic AMP -- metabolism
- DNA, Complementary -- genetics
- Dose-Response Relationship, Drug
- Humans
- In Vitro Techniques
- Indoles -- metabolism
- Ligands
- Morpholines -- metabolism
- Mutagenesis
- Naphthalenes -- metabolism
- Plasmids
- Protein Binding
- Receptors, Cannabinoid
- Receptors, Drug -- chemistry
- Recombinant Fusion Proteins -- metabolism
- Spleen -- physiology
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
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