Grapefruit juice activates P-glycoprotein-mediated drug transport. [electronic resource]
Producer: 19990625Description: 478-85 p. digitalISSN:- 0724-8741
- ATP Binding Cassette Transporter, Subfamily B, Member 1 -- metabolism
- Animals
- Antineoplastic Agents, Phytogenic -- pharmacokinetics
- Aryl Hydrocarbon Hydroxylases
- Beverages
- Biological Availability
- Biological Transport, Active
- Caco-2 Cells -- metabolism
- Cells, Cultured
- Citrus
- Cytochrome P-450 CYP3A
- Cytochrome P-450 Enzyme Inhibitors
- Cytochrome P-450 Enzyme System -- metabolism
- Diuretics, Osmotic -- pharmacokinetics
- Dogs
- Humans
- Kidney -- cytology
- Mannitol -- pharmacokinetics
- Oxidoreductases, N-Demethylating -- antagonists & inhibitors
- Pharmacokinetics
- Vinblastine -- pharmacokinetics
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
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