Synthesis, CoMFA analysis, and receptor docking of 3,5-diacyl-2, 4-dialkylpyridine derivatives as selective A3 adenosine receptor antagonists. [electronic resource]
Producer: 19990316Description: 706-21 p. digitalISSN:- 0022-2623
- Animals
- Binding Sites
- Binding, Competitive
- Bridged Bicyclo Compounds, Heterocyclic -- chemical synthesis
- CHO Cells
- Cell Line
- Cerebral Cortex -- metabolism
- Cricetinae
- Humans
- In Vitro Techniques
- Ligands
- Mice
- Models, Molecular
- Neostriatum -- metabolism
- Purinergic P1 Receptor Agonists
- Radioligand Assay
- Rats
- Receptor, Adenosine A3
- Receptors, Purinergic P1 -- metabolism
- Recombinant Proteins -- agonists
- Structure-Activity Relationship
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Publication Type: Journal Article
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