BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability. (Record no. 28406472)
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| 000 -LEADER | |
|---|---|
| fixed length control field | 02145 a2200649 4500 |
| 005 - DATE AND TIME OF LATEST TRANSACTION | |
| control field | 20250517215354.0 |
| 008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
| fixed length control field | 201812s 0 0 eng d |
| 022 ## - INTERNATIONAL STANDARD SERIAL NUMBER | |
| International Standard Serial Number | 1464-3391 |
| 024 7# - OTHER STANDARD IDENTIFIER | |
| Standard number or code | 10.1016/j.bmc.2018.05.003 |
| Source of number or code | doi |
| 040 ## - CATALOGING SOURCE | |
| Original cataloging agency | NLM |
| Language of cataloging | eng |
| Transcribing agency | NLM |
| 100 1# - MAIN ENTRY--PERSONAL NAME | |
| Personal name | Jennings, Laura E |
| 264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE | |
| Date of production, publication, distribution, manufacture, or copyright notice | 20181227 |
| 245 00 - TITLE STATEMENT | |
| Title | BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability. |
| Medium | [electronic resource] |
| 260 ## - PUBLICATION, DISTRIBUTION, ETC. | |
| Name of publisher, distributor, etc. | Bioorganic & medicinal chemistry |
| Date of publication, distribution, etc. | 07 2018 |
| 300 ## - PHYSICAL DESCRIPTION | |
| Extent | 2937-2957 p. |
| Other physical details | digital |
| 500 ## - GENERAL NOTE | |
| General note | Publication Type: Journal Article; Research Support, Non-U.S. Gov't |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Biological Assay |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Blotting, Western |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Cell Cycle Proteins |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Crystallography, X-Ray |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Drug Stability |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Heterocyclic Compounds, 4 or More Rings |
| General subdivision | chemistry |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Humans |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Inhibitory Concentration 50 |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Ligands |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Luciferases |
| General subdivision | chemistry |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | MCF-7 Cells |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Molecular Dynamics Simulation |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Molecular Structure |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Nuclear Proteins |
| General subdivision | chemistry |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Structure-Activity Relationship |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Transcription Factors |
| General subdivision | chemistry |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Schiedel, Matthias |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Hewings, David S |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Picaud, Sarah |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Laurin, Corentine M C |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Bruno, Paul A |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Bluck, Joseph P |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Scorah, Amy R |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | See, Larissa |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Reynolds, Jessica K |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Moroglu, Mustafa |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Mistry, Ishna N |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Hicks, Amy |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Guzanov, Pavel |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Clayton, James |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Evans, Charles N G |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Stazi, Giulia |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Biggin, Philip C |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Mapp, Anna K |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Hammond, Ester M |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Humphreys, Philip G |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Filippakopoulos, Panagis |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Conway, Stuart J |
| 773 0# - HOST ITEM ENTRY | |
| Title | Bioorganic & medicinal chemistry |
| Related parts | vol. 26 |
| -- | no. 11 |
| -- | p. 2937-2957 |
| 856 40 - ELECTRONIC LOCATION AND ACCESS | |
| Uniform Resource Identifier | <a href="https://doi.org/10.1016/j.bmc.2018.05.003">https://doi.org/10.1016/j.bmc.2018.05.003</a> |
| Public note | Available from publisher's website |
No items available.