Discovery, Structure-Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors. (Record no. 27390846)

MARC details
000 -LEADER
fixed length control field 02447 a2200757 4500
005 - DATE AND TIME OF LATEST TRANSACTION
control field 20250517164231.0
008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION
fixed length control field 201709s 0 0 eng d
022 ## - INTERNATIONAL STANDARD SERIAL NUMBER
International Standard Serial Number 1520-4804
024 7# - OTHER STANDARD IDENTIFIER
Standard number or code 10.1021/acs.jmedchem.7b00647
Source of number or code doi
040 ## - CATALOGING SOURCE
Original cataloging agency NLM
Language of cataloging eng
Transcribing agency NLM
100 1# - MAIN ENTRY--PERSONAL NAME
Personal name Joncour, Agnès
264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE
Date of production, publication, distribution, manufacture, or copyright notice 20170926
245 00 - TITLE STATEMENT
Title Discovery, Structure-Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors.
Medium [electronic resource]
260 ## - PUBLICATION, DISTRIBUTION, ETC.
Name of publisher, distributor, etc. Journal of medicinal chemistry
Date of publication, distribution, etc. 09 2017
300 ## - PHYSICAL DESCRIPTION
Extent 7371-7392 p.
Other physical details digital
500 ## - GENERAL NOTE
General note Publication Type: Journal Article; Research Support, Non-U.S. Gov't
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Animals
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Humans
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Imidazoles
General subdivision chemistry
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Lysophosphatidylcholines
General subdivision metabolism
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Lysophospholipids
General subdivision metabolism
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Male
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Mice
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Molecular Docking Simulation
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Phosphodiesterase Inhibitors
General subdivision chemistry
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Phosphoric Diester Hydrolases
General subdivision chemistry
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Pyridines
General subdivision chemistry
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Rats
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Rats, Sprague-Dawley
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM
Topical term or geographic name entry element Structure-Activity Relationship
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Desroy, Nicolas
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Housseman, Christopher
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Bock, Xavier
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Bienvenu, Natacha
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Cherel, Laëtitia
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Labeguere, Virginie
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Peixoto, Christophe
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Annoot, Denis
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Lepissier, Luce
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Heiermann, Jörg
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Hengeveld, Willem Jan
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Pilzak, Gregor
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Monjardet, Alain
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Wakselman, Emanuelle
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Roncoroni, Veronique
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Le Tallec, Sandrine
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Galien, René
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name David, Christelle
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Vandervoort, Nele
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Christophe, Thierry
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Conrath, Katja
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Jans, Mia
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Wohlkonig, Alexandre
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Soror, Sameh
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Steyaert, Jan
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Touitou, Robert
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Fleury, Damien
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Vercheval, Lionel
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Mollat, Patrick
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Triballeau, Nicolas
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name van der Aar, Ellen
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Brys, Reginald
700 1# - ADDED ENTRY--PERSONAL NAME
Personal name Heckmann, Bertrand
773 0# - HOST ITEM ENTRY
Title Journal of medicinal chemistry
Related parts vol. 60
-- no. 17
-- p. 7371-7392
856 40 - ELECTRONIC LOCATION AND ACCESS
Uniform Resource Identifier <a href="https://doi.org/10.1021/acs.jmedchem.7b00647">https://doi.org/10.1021/acs.jmedchem.7b00647</a>
Public note Available from publisher's website

No items available.