BI 1002494, a Novel Potent and Selective Oral Spleen Tyrosine Kinase Inhibitor, Displays Differential Potency in Human Basophils and B Cells. (Record no. 25896792)
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000 -LEADER | |
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fixed length control field | 02341 a2200697 4500 |
005 - DATE AND TIME OF LATEST TRANSACTION | |
control field | 20250517090707.0 |
008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
fixed length control field | 201705s 0 0 eng d |
022 ## - INTERNATIONAL STANDARD SERIAL NUMBER | |
International Standard Serial Number | 1521-0103 |
024 7# - OTHER STANDARD IDENTIFIER | |
Standard number or code | 10.1124/jpet.116.233155 |
Source of number or code | doi |
040 ## - CATALOGING SOURCE | |
Original cataloging agency | NLM |
Language of cataloging | eng |
Transcribing agency | NLM |
100 1# - MAIN ENTRY--PERSONAL NAME | |
Personal name | Lamb, David J |
264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE | |
Date of production, publication, distribution, manufacture, or copyright notice | 20170523 |
245 00 - TITLE STATEMENT | |
Title | BI 1002494, a Novel Potent and Selective Oral Spleen Tyrosine Kinase Inhibitor, Displays Differential Potency in Human Basophils and B Cells. |
Medium | [electronic resource] |
260 ## - PUBLICATION, DISTRIBUTION, ETC. | |
Name of publisher, distributor, etc. | The Journal of pharmacology and experimental therapeutics |
Date of publication, distribution, etc. | 06 2016 |
300 ## - PHYSICAL DESCRIPTION | |
Extent | 554-61 p. |
Other physical details | digital |
500 ## - GENERAL NOTE | |
General note | Publication Type: Journal Article; Research Support, Non-U.S. Gov't |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Administration, Oral |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Animals |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | B-Lymphocytes |
General subdivision | drug effects |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Basophils |
General subdivision | drug effects |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Humans |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Male |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Mast Cells |
General subdivision | drug effects |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Naphthyridines |
General subdivision | administration & dosage |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Protein Kinase Inhibitors |
General subdivision | administration & dosage |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Pyrrolidines |
General subdivision | administration & dosage |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Pyrrolidinones |
General subdivision | administration & dosage |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Rats |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Syk Kinase |
General subdivision | antagonists & inhibitors |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Wollin, Stefan Lutz |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Schnapp, Andreas |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Bischoff, Daniel |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Erb, Klaus J |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Bouyssou, Thierry |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Guilliard, Bernd |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Strasser, Christine |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Wex, Eva |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Blum, Sylvia |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Thaler, Eva |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Nickel, Helga |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Radmacher, Oliver |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Haas, Hannah |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Swantek, Jennifer L |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Souza, Don |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Canfield, Melissa |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | White, Della |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Panzenbeck, Mark |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Kashem, Mohammed A |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Sanville-Ross, Mary |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Kono, Takeshi |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Sewald, Katherina |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Braun, Armin |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Obernolte, Helena |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Danov, Olga |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Schaenzle, Gerhard |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Rast, Georg |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Maier, Gerd-Michael |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Hoffmann, Matthias |
773 0# - HOST ITEM ENTRY | |
Title | The Journal of pharmacology and experimental therapeutics |
Related parts | vol. 357 |
-- | no. 3 |
-- | p. 554-61 |
856 40 - ELECTRONIC LOCATION AND ACCESS | |
Uniform Resource Identifier | <a href="https://doi.org/10.1124/jpet.116.233155">https://doi.org/10.1124/jpet.116.233155</a> |
Public note | Available from publisher's website |
No items available.