Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach. (Record no. 25170804)
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fixed length control field | 02493 a2200769 4500 |
005 - DATE AND TIME OF LATEST TRANSACTION | |
control field | 20250517045639.0 |
008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
fixed length control field | 201512s 0 0 eng d |
022 ## - INTERNATIONAL STANDARD SERIAL NUMBER | |
International Standard Serial Number | 1520-4804 |
024 7# - OTHER STANDARD IDENTIFIER | |
Standard number or code | 10.1021/acs.jmedchem.5b01082 |
Source of number or code | doi |
040 ## - CATALOGING SOURCE | |
Original cataloging agency | NLM |
Language of cataloging | eng |
Transcribing agency | NLM |
100 1# - MAIN ENTRY--PERSONAL NAME | |
Personal name | Engel, Julian |
264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE | |
Date of production, publication, distribution, manufacture, or copyright notice | 20151214 |
245 00 - TITLE STATEMENT | |
Title | Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach. |
Medium | [electronic resource] |
260 ## - PUBLICATION, DISTRIBUTION, ETC. | |
Name of publisher, distributor, etc. | Journal of medicinal chemistry |
Date of publication, distribution, etc. | Sep 2015 |
300 ## - PHYSICAL DESCRIPTION | |
Extent | 6844-63 p. |
Other physical details | digital |
500 ## - GENERAL NOTE | |
General note | Publication Type: Journal Article; Research Support, Non-U.S. Gov't |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Antineoplastic Agents |
General subdivision | chemistry |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Carcinoma, Non-Small-Cell Lung |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Cell Line, Tumor |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Cell Membrane Permeability |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Crystallography, X-Ray |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Databases, Chemical |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Drug Design |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Drug Resistance, Neoplasm |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | ErbB Receptors |
General subdivision | antagonists & inhibitors |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Humans |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Kinetics |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Lung Neoplasms |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Models, Molecular |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Molecular Conformation |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Mutation |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Pyrazoles |
General subdivision | chemistry |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Pyrimidines |
General subdivision | chemistry |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Quinazolines |
General subdivision | chemistry |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Small Molecule Libraries |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Solubility |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Structure-Activity Relationship |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | src-Family Kinases |
General subdivision | chemistry |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Richters, André |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Getlik, Matthäus |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Tomassi, Stefano |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Keul, Marina |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Termathe, Martin |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Lategahn, Jonas |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Becker, Christian |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Mayer-Wrangowski, Svenja |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Grütter, Christian |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Uhlenbrock, Niklas |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Krüll, Jasmin |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Schaumann, Niklas |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Eppmann, Simone |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Kibies, Patrick |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Hoffgaard, Franziska |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Heil, Jochen |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Menninger, Sascha |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Ortiz-Cuaran, Sandra |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Heuckmann, Johannes M |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Tinnefeld, Verena |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Zahedi, René P |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Sos, Martin L |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Schultz-Fademrecht, Carsten |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Thomas, Roman K |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Kast, Stefan M |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Rauh, Daniel |
773 0# - HOST ITEM ENTRY | |
Title | Journal of medicinal chemistry |
Related parts | vol. 58 |
-- | no. 17 |
-- | p. 6844-63 |
856 40 - ELECTRONIC LOCATION AND ACCESS | |
Uniform Resource Identifier | <a href="https://doi.org/10.1021/acs.jmedchem.5b01082">https://doi.org/10.1021/acs.jmedchem.5b01082</a> |
Public note | Available from publisher's website |
No items available.