Lead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists. (Record no. 22164281)
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| 000 -LEADER | |
|---|---|
| fixed length control field | 01771 a2200541 4500 |
| 005 - DATE AND TIME OF LATEST TRANSACTION | |
| control field | 20250516114151.0 |
| 008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
| fixed length control field | 201304s 0 0 eng d |
| 022 ## - INTERNATIONAL STANDARD SERIAL NUMBER | |
| International Standard Serial Number | 1860-7187 |
| 024 7# - OTHER STANDARD IDENTIFIER | |
| Standard number or code | 10.1002/cmdc.201200406 |
| Source of number or code | doi |
| 040 ## - CATALOGING SOURCE | |
| Original cataloging agency | NLM |
| Language of cataloging | eng |
| Transcribing agency | NLM |
| 100 1# - MAIN ENTRY--PERSONAL NAME | |
| Personal name | Provins, Laurent |
| 264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE | |
| Date of production, publication, distribution, manufacture, or copyright notice | 20130429 |
| 245 00 - TITLE STATEMENT | |
| Title | Lead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists. |
| Medium | [electronic resource] |
| 260 ## - PUBLICATION, DISTRIBUTION, ETC. | |
| Name of publisher, distributor, etc. | ChemMedChem |
| Date of publication, distribution, etc. | Dec 2012 |
| 300 ## - PHYSICAL DESCRIPTION | |
| Extent | 2087-92 p. |
| Other physical details | digital |
| 500 ## - GENERAL NOTE | |
| General note | Publication Type: Journal Article; Research Support, Non-U.S. Gov't |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Animals |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Benzamides |
| General subdivision | chemistry |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Caco-2 Cells |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Histamine Agonists |
| General subdivision | chemistry |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Humans |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Male |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Piperidines |
| General subdivision | chemistry |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Rats |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Rats, Wistar |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Receptors, Histamine H3 |
| General subdivision | metabolism |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Structure-Activity Relationship |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Thiazoles |
| General subdivision | chemistry |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Trans-Activators |
| General subdivision | metabolism |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Transcriptional Regulator ERG |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Denonne, Frédéric |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Célanire, Sylvain |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Christophe, Bernard |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Defays, Sabine |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Delaunoy, Christel |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Delporte, Marie-Laure |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Demaude, Thierry |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Durieu, Véronique |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Gillard, Michel |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Hubert, Delphine |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Lamberty, Yves |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Lorent, Geneviève |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Valade, Anne |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Vanbellinghen, Alain |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Van Houtvin, Nathalie |
| 773 0# - HOST ITEM ENTRY | |
| Title | ChemMedChem |
| Related parts | vol. 7 |
| -- | no. 12 |
| -- | p. 2087-92 |
| 856 40 - ELECTRONIC LOCATION AND ACCESS | |
| Uniform Resource Identifier | <a href="https://doi.org/10.1002/cmdc.201200406">https://doi.org/10.1002/cmdc.201200406</a> |
| Public note | Available from publisher's website |
No items available.