Azepanone-based inhibitors of human cathepsin S: optimization of selectivity via the P2 substituent. (Record no. 20986117)
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| 000 -LEADER | |
|---|---|
| fixed length control field | 01783 a2200505 4500 |
| 005 - DATE AND TIME OF LATEST TRANSACTION | |
| control field | 20250516044613.0 |
| 008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
| fixed length control field | 201111s 0 0 eng d |
| 022 ## - INTERNATIONAL STANDARD SERIAL NUMBER | |
| International Standard Serial Number | 1464-3405 |
| 024 7# - OTHER STANDARD IDENTIFIER | |
| Standard number or code | 10.1016/j.bmcl.2011.06.045 |
| Source of number or code | doi |
| 040 ## - CATALOGING SOURCE | |
| Original cataloging agency | NLM |
| Language of cataloging | eng |
| Transcribing agency | NLM |
| 100 1# - MAIN ENTRY--PERSONAL NAME | |
| Personal name | Kerns, Jeffrey K |
| 264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE | |
| Date of production, publication, distribution, manufacture, or copyright notice | 20111122 |
| 245 00 - TITLE STATEMENT | |
| Title | Azepanone-based inhibitors of human cathepsin S: optimization of selectivity via the P2 substituent. |
| Medium | [electronic resource] |
| 260 ## - PUBLICATION, DISTRIBUTION, ETC. | |
| Name of publisher, distributor, etc. | Bioorganic & medicinal chemistry letters |
| Date of publication, distribution, etc. | Aug 2011 |
| 300 ## - PHYSICAL DESCRIPTION | |
| Extent | 4409-15 p. |
| Other physical details | digital |
| 500 ## - GENERAL NOTE | |
| General note | Publication Type: Journal Article; Research Support, Non-U.S. Gov't |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Alanine |
| General subdivision | chemistry |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Azepines |
| General subdivision | chemical synthesis |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Binding Sites |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Cathepsin K |
| General subdivision | antagonists & inhibitors |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Cathepsin L |
| General subdivision | antagonists & inhibitors |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Cathepsins |
| General subdivision | antagonists & inhibitors |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Computer Simulation |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Humans |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Niacinamide |
| General subdivision | analogs & derivatives |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Protease Inhibitors |
| General subdivision | chemical synthesis |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Stereoisomerism |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Structure-Activity Relationship |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Nie, Hong |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Bondinell, William |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Widdowson, Katherine L |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Yamashita, Dennis S |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Rahman, Attiq |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Podolin, Patricia L |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Carpenter, Donald C |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Jin, Qi |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Riflade, Benoit |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Dong, Xiaoyang |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Nevins, Neysa |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Keller, Paul M |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Mitchell, Laura |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Tomaszek, Thaddeus |
| 773 0# - HOST ITEM ENTRY | |
| Title | Bioorganic & medicinal chemistry letters |
| Related parts | vol. 21 |
| -- | no. 15 |
| -- | p. 4409-15 |
| 856 40 - ELECTRONIC LOCATION AND ACCESS | |
| Uniform Resource Identifier | <a href="https://doi.org/10.1016/j.bmcl.2011.06.045">https://doi.org/10.1016/j.bmcl.2011.06.045</a> |
| Public note | Available from publisher's website |
No items available.