Discovery of INCB10820/PF-4178903, a potent, selective, and orally bioavailable dual CCR2 and CCR5 antagonist. (Record no. 20573919)
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| 000 -LEADER | |
|---|---|
| fixed length control field | 01995 a2200637 4500 |
| 005 - DATE AND TIME OF LATEST TRANSACTION | |
| control field | 20250516023021.0 |
| 008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
| fixed length control field | 201106s 0 0 eng d |
| 022 ## - INTERNATIONAL STANDARD SERIAL NUMBER | |
| International Standard Serial Number | 1464-3405 |
| 024 7# - OTHER STANDARD IDENTIFIER | |
| Standard number or code | 10.1016/j.bmcl.2011.01.015 |
| Source of number or code | doi |
| 040 ## - CATALOGING SOURCE | |
| Original cataloging agency | NLM |
| Language of cataloging | eng |
| Transcribing agency | NLM |
| 100 1# - MAIN ENTRY--PERSONAL NAME | |
| Personal name | Zheng, Changsheng |
| 264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE | |
| Date of production, publication, distribution, manufacture, or copyright notice | 20110614 |
| 245 00 - TITLE STATEMENT | |
| Title | Discovery of INCB10820/PF-4178903, a potent, selective, and orally bioavailable dual CCR2 and CCR5 antagonist. |
| Medium | [electronic resource] |
| 260 ## - PUBLICATION, DISTRIBUTION, ETC. | |
| Name of publisher, distributor, etc. | Bioorganic & medicinal chemistry letters |
| Date of publication, distribution, etc. | Mar 2011 |
| 300 ## - PHYSICAL DESCRIPTION | |
| Extent | 1442-6 p. |
| Other physical details | digital |
| 500 ## - GENERAL NOTE | |
| General note | Publication Type: Journal Article |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Biological Availability |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | CCR5 Receptor Antagonists |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Caco-2 Cells |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Drug Discovery |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Humans |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Inhibitory Concentration 50 |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Molecular Structure |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Piperazines |
| General subdivision | chemical synthesis |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Pyrans |
| General subdivision | chemical synthesis |
| 650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | Receptors, CCR2 |
| General subdivision | antagonists & inhibitors |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Cao, Ganfeng |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Xia, Michael |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Feng, Hao |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Glenn, Joseph |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Anand, Rajan |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Zhang, Ke |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Huang, Taisheng |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Wang, Anlai |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Kong, Ling |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Li, Mei |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Galya, Laurine |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Hughes, Robert O |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Devraj, Rajesh |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Morton, Phillip A |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Rogier, D Joseph |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Covington, Maryanne |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Baribaud, Fred |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Shin, Niu |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Scherle, Peggy |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Diamond, Sharon |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Yeleswaram, Swamy |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Vaddi, Kris |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Newton, Robert |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Hollis, Greg |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Friedman, Steven |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Metcalf, Brian |
| 700 1# - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Xue, Chu-Biao |
| 773 0# - HOST ITEM ENTRY | |
| Title | Bioorganic & medicinal chemistry letters |
| Related parts | vol. 21 |
| -- | no. 5 |
| -- | p. 1442-6 |
| 856 40 - ELECTRONIC LOCATION AND ACCESS | |
| Uniform Resource Identifier | <a href="https://doi.org/10.1016/j.bmcl.2011.01.015">https://doi.org/10.1016/j.bmcl.2011.01.015</a> |
| Public note | Available from publisher's website |
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