In vitro intrinsic clearance-based optimization of N3-phenylpyrazinones as corticotropin-releasing factor-1 (CRF1) receptor antagonists. (Record no. 18970039)
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fixed length control field | 01856 a2200577 4500 |
005 - DATE AND TIME OF LATEST TRANSACTION | |
control field | 20250515175129.0 |
008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
fixed length control field | 200908s 0 0 eng d |
022 ## - INTERNATIONAL STANDARD SERIAL NUMBER | |
International Standard Serial Number | 1520-4804 |
024 7# - OTHER STANDARD IDENTIFIER | |
Standard number or code | 10.1021/jm900302q |
Source of number or code | doi |
040 ## - CATALOGING SOURCE | |
Original cataloging agency | NLM |
Language of cataloging | eng |
Transcribing agency | NLM |
100 1# - MAIN ENTRY--PERSONAL NAME | |
Personal name | Hartz, Richard A |
264 #0 - PRODUCTION, PUBLICATION, DISTRIBUTION, MANUFACTURE, AND COPYRIGHT NOTICE | |
Date of production, publication, distribution, manufacture, or copyright notice | 20090825 |
245 00 - TITLE STATEMENT | |
Title | In vitro intrinsic clearance-based optimization of N3-phenylpyrazinones as corticotropin-releasing factor-1 (CRF1) receptor antagonists. |
Medium | [electronic resource] |
260 ## - PUBLICATION, DISTRIBUTION, ETC. | |
Name of publisher, distributor, etc. | Journal of medicinal chemistry |
Date of publication, distribution, etc. | Jul 2009 |
300 ## - PHYSICAL DESCRIPTION | |
Extent | 4161-72 p. |
Other physical details | digital |
500 ## - GENERAL NOTE | |
General note | Publication Type: Journal Article |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Animals |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Humans |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Inhibitory Concentration 50 |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Male |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Metabolic Clearance Rate |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Pyrazines |
General subdivision | chemistry |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Rats |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | Receptors, Corticotropin-Releasing Hormone |
General subdivision | antagonists & inhibitors |
650 04 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
Topical term or geographic name entry element | CRF Receptor, Type 1 |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Ahuja, Vijay T |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Rafalski, Maria |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Schmitz, William D |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Brenner, Allison B |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Denhart, Derek J |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Ditta, Jonathan L |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Deskus, Jeffrey A |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Yue, Eddy W |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Arvanitis, Argyrios G |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Lelas, Snjezana |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Li, Yu-Wen |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Molski, Thaddeus F |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Wong, Harvey |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Grace, James E |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Lentz, Kimberley A |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Li, Jianqing |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Lodge, Nicholas J |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Zaczek, Robert |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Combs, Andrew P |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Olson, Richard E |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Mattson, Ronald J |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Bronson, Joanne J |
700 1# - ADDED ENTRY--PERSONAL NAME | |
Personal name | Macor, John E |
773 0# - HOST ITEM ENTRY | |
Title | Journal of medicinal chemistry |
Related parts | vol. 52 |
-- | no. 14 |
-- | p. 4161-72 |
856 40 - ELECTRONIC LOCATION AND ACCESS | |
Uniform Resource Identifier | <a href="https://doi.org/10.1021/jm900302q">https://doi.org/10.1021/jm900302q</a> |
Public note | Available from publisher's website |
No items available.