Potent piperazine hydroxyethylamine HIV protease inhibitors containing novel P3 ligands.

Chen, X

Potent piperazine hydroxyethylamine HIV protease inhibitors containing novel P3 ligands. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 1998 - 3531-6 p. digital

Publication Type: Journal Article

0960-894X

10.1016/s0960-894x(98)00653-2 doi


Animals
Anti-HIV Agents--chemical synthesis
Blood
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme Inhibitors
HIV--drug effects
HIV Protease Inhibitors--chemical synthesis
Humans
Ligands
Microbial Sensitivity Tests
Microsomes, Liver--enzymology
Mixed Function Oxygenases--antagonists & inhibitors
Piperazines--chemical synthesis