Potent piperazine hydroxyethylamine HIV protease inhibitors containing novel P3 ligands.
Chen, X
Potent piperazine hydroxyethylamine HIV protease inhibitors containing novel P3 ligands. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 1998 - 3531-6 p. digital
Publication Type: Journal Article
0960-894X
10.1016/s0960-894x(98)00653-2 doi
Animals
Anti-HIV Agents--chemical synthesis
Blood
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme Inhibitors
HIV--drug effects
HIV Protease Inhibitors--chemical synthesis
Humans
Ligands
Microbial Sensitivity Tests
Microsomes, Liver--enzymology
Mixed Function Oxygenases--antagonists & inhibitors
Piperazines--chemical synthesis
Potent piperazine hydroxyethylamine HIV protease inhibitors containing novel P3 ligands. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 1998 - 3531-6 p. digital
Publication Type: Journal Article
0960-894X
10.1016/s0960-894x(98)00653-2 doi
Animals
Anti-HIV Agents--chemical synthesis
Blood
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme Inhibitors
HIV--drug effects
HIV Protease Inhibitors--chemical synthesis
Humans
Ligands
Microbial Sensitivity Tests
Microsomes, Liver--enzymology
Mixed Function Oxygenases--antagonists & inhibitors
Piperazines--chemical synthesis