Potent and selective bicyclic lactam inhibitors of thrombin: Part 2: P1 modifications.
Plummer, J S
Potent and selective bicyclic lactam inhibitors of thrombin: Part 2: P1 modifications. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 1998 - 3409-14 p. digital
Publication Type: Journal Article
0960-894X
10.1016/s0960-894x(98)00613-1 doi
Animals
Fibrinolytic Agents--chemical synthesis
Lactams--chemical synthesis
Rats
Serine Proteinase Inhibitors--chemical synthesis
Structure-Activity Relationship
Thrombin--antagonists & inhibitors
Potent and selective bicyclic lactam inhibitors of thrombin: Part 2: P1 modifications. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 1998 - 3409-14 p. digital
Publication Type: Journal Article
0960-894X
10.1016/s0960-894x(98)00613-1 doi
Animals
Fibrinolytic Agents--chemical synthesis
Lactams--chemical synthesis
Rats
Serine Proteinase Inhibitors--chemical synthesis
Structure-Activity Relationship
Thrombin--antagonists & inhibitors