In vitro inhibition of hepadnavirus polymerases by the triphosphates of BMS-200475 and lobucavir.

Seifer, M

In vitro inhibition of hepadnavirus polymerases by the triphosphates of BMS-200475 and lobucavir. [electronic resource] - Antimicrobial agents and chemotherapy Dec 1998 - 3200-8 p. digital

Publication Type: Journal Article

0066-4804

10.1128/AAC.42.12.3200 doi


Antiviral Agents--pharmacology
DNA-Directed RNA Polymerases--antagonists & inhibitors
Deoxyguanosine--analogs & derivatives
Enzyme Inhibitors--pharmacology
Guanine--analogs & derivatives
Hepadnaviridae--enzymology
Hepatitis B Virus, Duck--drug effects
Hepatitis B Virus, Woodchuck--drug effects
Hepatitis B virus--drug effects
Humans
Kinetics
Nucleic Acid Synthesis Inhibitors
Phosphates
RNA-Directed DNA Polymerase--metabolism
Structure-Activity Relationship