Ligand efficacy and potency at recombinant alpha2 adrenergic receptors: agonist-mediated [35S]GTPgammaS binding.
Jasper, J R
Ligand efficacy and potency at recombinant alpha2 adrenergic receptors: agonist-mediated [35S]GTPgammaS binding. [electronic resource] - Biochemical pharmacology Apr 1998 - 1035-43 p. digital
Publication Type: Journal Article
0006-2952
10.1016/s0006-2952(97)00631-x doi
Adenylyl Cyclases--metabolism
Adrenergic alpha-2 Receptor Agonists
Adrenergic alpha-Agonists--pharmacology
Adrenergic alpha-Antagonists--metabolism
Animals
Cell Line
Cell Membrane--metabolism
Cyclic AMP--metabolism
Genetic Vectors
Guanosine 5'-O-(3-Thiotriphosphate)--pharmacology
Humans
Ligands
Mice
Protein Binding
Quinolizines--metabolism
Radioligand Assay
Receptors, Adrenergic, alpha-2--chemistry
Recombinant Proteins--chemistry
Ligand efficacy and potency at recombinant alpha2 adrenergic receptors: agonist-mediated [35S]GTPgammaS binding. [electronic resource] - Biochemical pharmacology Apr 1998 - 1035-43 p. digital
Publication Type: Journal Article
0006-2952
10.1016/s0006-2952(97)00631-x doi
Adenylyl Cyclases--metabolism
Adrenergic alpha-2 Receptor Agonists
Adrenergic alpha-Agonists--pharmacology
Adrenergic alpha-Antagonists--metabolism
Animals
Cell Line
Cell Membrane--metabolism
Cyclic AMP--metabolism
Genetic Vectors
Guanosine 5'-O-(3-Thiotriphosphate)--pharmacology
Humans
Ligands
Mice
Protein Binding
Quinolizines--metabolism
Radioligand Assay
Receptors, Adrenergic, alpha-2--chemistry
Recombinant Proteins--chemistry