Characterization of [125I]-PD164333, an ETA selective non-peptide radiolabelled antagonist, in normal and diseased human tissues.
Davenport, A P
Characterization of [125I]-PD164333, an ETA selective non-peptide radiolabelled antagonist, in normal and diseased human tissues. [electronic resource] - British journal of pharmacology Jan 1998 - 223-30 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0007-1188
10.1038/sj.bjp.0701597 doi
Adult
Aorta--diagnostic imaging
Autoradiography
Brain--diagnostic imaging
Crotonates--metabolism
Dioxoles--metabolism
Drug Stability
Endothelin Receptor Antagonists
Endothelin-1--pharmacology
Female
Heart Ventricles--diagnostic imaging
Humans
Iodine Radioisotopes
Kidney--diagnostic imaging
Kinetics
Ligands
Male
Middle Aged
Radionuclide Imaging
Radiopharmaceuticals--metabolism
Receptor, Endothelin A
Receptors, Endothelin--metabolism
Characterization of [125I]-PD164333, an ETA selective non-peptide radiolabelled antagonist, in normal and diseased human tissues. [electronic resource] - British journal of pharmacology Jan 1998 - 223-30 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0007-1188
10.1038/sj.bjp.0701597 doi
Adult
Aorta--diagnostic imaging
Autoradiography
Brain--diagnostic imaging
Crotonates--metabolism
Dioxoles--metabolism
Drug Stability
Endothelin Receptor Antagonists
Endothelin-1--pharmacology
Female
Heart Ventricles--diagnostic imaging
Humans
Iodine Radioisotopes
Kidney--diagnostic imaging
Kinetics
Ligands
Male
Middle Aged
Radionuclide Imaging
Radiopharmaceuticals--metabolism
Receptor, Endothelin A
Receptors, Endothelin--metabolism