Evaluation in rat of RS-79948-197 as a potential PET ligand for central alpha 2-adrenoceptors.

Hume, S P

Evaluation in rat of RS-79948-197 as a potential PET ligand for central alpha 2-adrenoceptors. [electronic resource] - European journal of pharmacology Dec 1996 - 67-73 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0014-2999

10.1016/s0014-2999(96)00710-8 doi


Adrenergic alpha-2 Receptor Antagonists
Adrenergic alpha-Antagonists--pharmacology
Animals
Brain--anatomy & histology
Imidazoline Receptors
Injections, Intravenous
Isoquinolines--pharmacokinetics
Ligands
Male
Naphthyridines--pharmacokinetics
Piperazines--pharmacology
Pyridines--pharmacology
Rats
Rats, Sprague-Dawley
Receptors, Adrenergic, alpha-2--drug effects
Receptors, Drug--antagonists & inhibitors
Serotonin Antagonists--pharmacology
Tissue Distribution
Tomography, Emission-Computed--methods