GR205171: a novel antagonist with high affinity for the tachykinin NK1 receptor, and potent broad-spectrum anti-emetic activity.
Gardner, C J
GR205171: a novel antagonist with high affinity for the tachykinin NK1 receptor, and potent broad-spectrum anti-emetic activity. [electronic resource] - Regulatory peptides Aug 1996 - 45-53 p. digital
Publication Type: Journal Article
0167-0115
10.1016/0167-0115(96)00071-7 doi
Administration, Oral
Animals
Antiemetics--metabolism
Cisplatin--adverse effects
Dogs
Dose-Response Relationship, Drug
Ferrets
Humans
Male
Motor Activity
Neurokinin-1 Receptor Antagonists
Piperidines--metabolism
Receptors, Neurokinin-1--metabolism
Shrews
Stereoisomerism
Tetrazoles--metabolism
GR205171: a novel antagonist with high affinity for the tachykinin NK1 receptor, and potent broad-spectrum anti-emetic activity. [electronic resource] - Regulatory peptides Aug 1996 - 45-53 p. digital
Publication Type: Journal Article
0167-0115
10.1016/0167-0115(96)00071-7 doi
Administration, Oral
Animals
Antiemetics--metabolism
Cisplatin--adverse effects
Dogs
Dose-Response Relationship, Drug
Ferrets
Humans
Male
Motor Activity
Neurokinin-1 Receptor Antagonists
Piperidines--metabolism
Receptors, Neurokinin-1--metabolism
Shrews
Stereoisomerism
Tetrazoles--metabolism