Pharmacology of L-744,453, a novel nonpeptidyl endothelin antagonist.

Williams, D L

Pharmacology of L-744,453, a novel nonpeptidyl endothelin antagonist. [electronic resource] - Life sciences 1996 - 1149-57 p. digital

Publication Type: Comparative Study; Journal Article

0024-3205

10.1016/0024-3205(96)00073-2 doi


Animals
Biological Availability
Blood Pressure--drug effects
CHO Cells--drug effects
Cricetinae
Dioxoles--metabolism
Dogs
Endothelin Receptor Antagonists
Endothelins--antagonists & inhibitors
Female
Ferrets
Humans
Hydrolysis
Imidazoles--metabolism
In Vitro Techniques
Iodine Radioisotopes
Kinetics
Male
Mice
Muscle Contraction--drug effects
Phosphatidylinositols--metabolism
Rats
Rats, Sprague-Dawley
Receptors, Endothelin--metabolism
Structure-Activity Relationship