Inhibition of the nicotinic acetylcholine receptor by barbiturates and by procaine: do they act at different sites?
Yost, C S
Inhibition of the nicotinic acetylcholine receptor by barbiturates and by procaine: do they act at different sites? [electronic resource] - Cellular and molecular neurobiology Apr 1993 - 159-72 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
0272-4340
10.1007/BF00735372 doi
Allosteric Site
Amino Acid Sequence
Amobarbital--pharmacology
Animals
Barbiturates--pharmacology
Binding Sites
Dimethylphenylpiperazinium Iodide--pharmacology
Dose-Response Relationship, Drug
Ion Channel Gating--drug effects
Membrane Potentials--drug effects
Mice
Molecular Sequence Data
Nicotinic Antagonists
Oocytes
Pentobarbital--pharmacology
Procaine--pharmacology
Protein Binding
Receptors, Nicotinic--genetics
Recombinant Proteins--antagonists & inhibitors
Secobarbital--pharmacology
Sodium Channels--drug effects
Xenopus laevis
Inhibition of the nicotinic acetylcholine receptor by barbiturates and by procaine: do they act at different sites? [electronic resource] - Cellular and molecular neurobiology Apr 1993 - 159-72 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
0272-4340
10.1007/BF00735372 doi
Allosteric Site
Amino Acid Sequence
Amobarbital--pharmacology
Animals
Barbiturates--pharmacology
Binding Sites
Dimethylphenylpiperazinium Iodide--pharmacology
Dose-Response Relationship, Drug
Ion Channel Gating--drug effects
Membrane Potentials--drug effects
Mice
Molecular Sequence Data
Nicotinic Antagonists
Oocytes
Pentobarbital--pharmacology
Procaine--pharmacology
Protein Binding
Receptors, Nicotinic--genetics
Recombinant Proteins--antagonists & inhibitors
Secobarbital--pharmacology
Sodium Channels--drug effects
Xenopus laevis