Probes for narcotic receptor mediated phenomena. 7. Synthesis and pharmacological properties of irreversible ligands specific for mu or delta opiate receptors.

Burke, T R

Probes for narcotic receptor mediated phenomena. 7. Synthesis and pharmacological properties of irreversible ligands specific for mu or delta opiate receptors. [electronic resource] - Journal of medicinal chemistry Dec 1984 - 1570-4 p. digital

Publication Type: Comparative Study; Journal Article

0022-2623

10.1021/jm00378a008 doi


Animals
Benzimidazoles--analogs & derivatives
Cell Line
Cell Membrane--metabolism
Chemical Phenomena
Chemistry
Drug Evaluation, Preclinical
Fentanyl--analogs & derivatives
Glioma--metabolism
Hybrid Cells--metabolism
Indicators and Reagents
Ligands--metabolism
Magnetic Resonance Spectroscopy
Mass Spectrometry
Mice
Narcotic Antagonists--chemical synthesis
Neuroblastoma--metabolism
Rats
Receptors, Opioid--drug effects
Receptors, Opioid, delta
Receptors, Opioid, mu
Structure-Activity Relationship
Thebaine--analogs & derivatives