Cholecystokinin antagonists. Synthesis of asperlicin analogues with improved potency and water solubility.

Bock, M G

Cholecystokinin antagonists. Synthesis of asperlicin analogues with improved potency and water solubility. [electronic resource] - Journal of medicinal chemistry Oct 1986 - 1941-5 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm00160a024 doi


Animals
Benzodiazepinones--chemical synthesis
Cholecystokinin--antagonists & inhibitors
Guinea Pigs
In Vitro Techniques
Rats
Receptors, Cholecystokinin--drug effects
Solubility
Structure-Activity Relationship