Discovery of novel TNNI3K inhibitor suppresses pyroptosis and apoptosis in murine myocardial infarction injury.
Pang, Haiying
Discovery of novel TNNI3K inhibitor suppresses pyroptosis and apoptosis in murine myocardial infarction injury. [electronic resource] - European journal of medicinal chemistry Jul 2020 - 112314 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2020.112314 doi
Animals
Apoptosis--drug effects
Binding Sites
Cardiotonic Agents--chemical synthesis
Cell Line
Drug Design
MAP Kinase Signaling System--drug effects
Male
Mice, Inbred C57BL
Molecular Docking Simulation
Molecular Structure
Myocardial Infarction--drug therapy
Protein Binding
Protein Kinase Inhibitors--chemical synthesis
Protein Serine-Threonine Kinases--antagonists & inhibitors
Pyroptosis--drug effects
Rats
Reactive Oxygen Species--metabolism
Structure-Activity Relationship
Discovery of novel TNNI3K inhibitor suppresses pyroptosis and apoptosis in murine myocardial infarction injury. [electronic resource] - European journal of medicinal chemistry Jul 2020 - 112314 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2020.112314 doi
Animals
Apoptosis--drug effects
Binding Sites
Cardiotonic Agents--chemical synthesis
Cell Line
Drug Design
MAP Kinase Signaling System--drug effects
Male
Mice, Inbred C57BL
Molecular Docking Simulation
Molecular Structure
Myocardial Infarction--drug therapy
Protein Binding
Protein Kinase Inhibitors--chemical synthesis
Protein Serine-Threonine Kinases--antagonists & inhibitors
Pyroptosis--drug effects
Rats
Reactive Oxygen Species--metabolism
Structure-Activity Relationship