Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to

Serafini, Marta

Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to [electronic resource] - Journal of medicinal chemistry 03 2020 - 3047-3065 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/acs.jmedchem.9b01809 doi


Animals
Benzimidazoles--blood
Cell Line, Tumor
Cells, Cultured
Enzyme Inhibitors--blood
Humans
Indoleamine-Pyrrole 2,3,-Dioxygenase--antagonists & inhibitors
Male
Mice
Molecular Docking Simulation
Structure-Activity Relationship