Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to
Serafini, Marta
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to [electronic resource] - Journal of medicinal chemistry 03 2020 - 3047-3065 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-4804
10.1021/acs.jmedchem.9b01809 doi
Animals
Benzimidazoles--blood
Cell Line, Tumor
Cells, Cultured
Enzyme Inhibitors--blood
Humans
Indoleamine-Pyrrole 2,3,-Dioxygenase--antagonists & inhibitors
Male
Mice
Molecular Docking Simulation
Structure-Activity Relationship
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to [electronic resource] - Journal of medicinal chemistry 03 2020 - 3047-3065 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-4804
10.1021/acs.jmedchem.9b01809 doi
Animals
Benzimidazoles--blood
Cell Line, Tumor
Cells, Cultured
Enzyme Inhibitors--blood
Humans
Indoleamine-Pyrrole 2,3,-Dioxygenase--antagonists & inhibitors
Male
Mice
Molecular Docking Simulation
Structure-Activity Relationship