Antibody-mediated delivery of chimeric protein degraders which target estrogen receptor alpha (ERα).

Dragovich, Peter S

Antibody-mediated delivery of chimeric protein degraders which target estrogen receptor alpha (ERα). [electronic resource] - Bioorganic & medicinal chemistry letters 02 2020 - 126907 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2019.126907 doi


Antibodies, Monoclonal--chemistry
Antineoplastic Agents--chemistry
Drug Carriers--chemistry
Drug Design
Estrogen Receptor alpha--immunology
Humans
Immunoconjugates--chemistry
MCF-7 Cells
Proteolysis--drug effects
Receptor, ErbB-2--metabolism