Structure-Based Design, Synthesis, and Biological Evaluation of Triazole-Based smHDAC8 Inhibitors.
Kalinin, Dmitrii V
Structure-Based Design, Synthesis, and Biological Evaluation of Triazole-Based smHDAC8 Inhibitors. [electronic resource] - ChemMedChem 04 2020 - 571-584 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1860-7187
10.1002/cmdc.201900583 doi
Animals
Drug Design
Histone Deacetylase Inhibitors--chemical synthesis
Histone Deacetylases--metabolism
Humans
Models, Molecular
Molecular Structure
Repressor Proteins--antagonists & inhibitors
Schistosoma mansoni--enzymology
Schistosomiasis--drug therapy
Triazoles--chemical synthesis
Structure-Based Design, Synthesis, and Biological Evaluation of Triazole-Based smHDAC8 Inhibitors. [electronic resource] - ChemMedChem 04 2020 - 571-584 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1860-7187
10.1002/cmdc.201900583 doi
Animals
Drug Design
Histone Deacetylase Inhibitors--chemical synthesis
Histone Deacetylases--metabolism
Humans
Models, Molecular
Molecular Structure
Repressor Proteins--antagonists & inhibitors
Schistosoma mansoni--enzymology
Schistosomiasis--drug therapy
Triazoles--chemical synthesis