Synthesis and Biological Evaluation of Structurally Diverse Benzimidazole Scaffolds as Potential Chemotherapeutic Agents.

Barasa, Leonard

Synthesis and Biological Evaluation of Structurally Diverse Benzimidazole Scaffolds as Potential Chemotherapeutic Agents. [electronic resource] - Anti-cancer agents in medicinal chemistry 2020 - 301-314 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1875-5992

10.2174/1871520619666191028101506 doi


A549 Cells
Amino Acids--chemistry
Anti-Bacterial Agents--chemical synthesis
Antineoplastic Agents--chemical synthesis
Apoptosis--drug effects
Benzimidazoles--chemical synthesis
DNA Topoisomerases--metabolism
Drug Evaluation, Preclinical
Escherichia coli--drug effects
Fatty Acids--chemistry
HeLa Cells
Hep G2 Cells
Humans
Indoles--chemistry
Microbial Sensitivity Tests
Staphylococcus aureus--drug effects
Staphylococcus epidermidis--drug effects
Structure-Activity Relationship
Topoisomerase Inhibitors--chemical synthesis