Biochemical and pharmacological characterization of an extremely potent and selective nonpeptide cholecystokinin antagonist.

Chang, R S

Biochemical and pharmacological characterization of an extremely potent and selective nonpeptide cholecystokinin antagonist. [electronic resource] - Proceedings of the National Academy of Sciences of the United States of America Jul 1986 - 4923-6 p. digital

Publication Type: Journal Article

0027-8424

10.1073/pnas.83.13.4923 doi


Animals
Benzodiazepines--antagonists & inhibitors
Benzodiazepinones--metabolism
Binding, Competitive
Brain--metabolism
Cattle
Cholecystokinin--antagonists & inhibitors
Devazepide
Gallbladder--metabolism
Gastric Mucosa--metabolism
Guinea Pigs
Ileum--drug effects
In Vitro Techniques
Membranes--metabolism
Muscle Contraction--drug effects
Pancreas--metabolism
Rats
Receptors, Cell Surface--metabolism
Receptors, Cholecystokinin