Synthesis and characterization of a high affinity radioiodinated probe for the alpha 2-adrenergic receptor.

Lanier, S M

Synthesis and characterization of a high affinity radioiodinated probe for the alpha 2-adrenergic receptor. [electronic resource] - Molecular pharmacology Mar 1986 - 219-27 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0026-895X


Animals
Binding, Competitive
Blood Platelets--metabolism
Calcium Channel Blockers--pharmacology
Chromatography, High Pressure Liquid
Epinephrine--metabolism
Humans
In Vitro Techniques
Iodine Radioisotopes
Kidney--metabolism
Kinetics
Ligands
Liver--metabolism
Male
Molecular Conformation
Norepinephrine--metabolism
Rats
Rats, Inbred Strains
Receptors, Adrenergic, alpha--metabolism
Secologanin Tryptamine Alkaloids--chemical synthesis
Structure-Activity Relationship
Yohimbine--metabolism