Selective inhibition of mutant IDH1 by DS-1001b ameliorates aberrant histone modifications and impairs tumor activity in chondrosarcoma.

Nakagawa, Makoto

Selective inhibition of mutant IDH1 by DS-1001b ameliorates aberrant histone modifications and impairs tumor activity in chondrosarcoma. [electronic resource] - Oncogene 10 2019 - 6835-6849 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1476-5594

10.1038/s41388-019-0929-9 doi


Bone Neoplasms--metabolism
Cell Cycle Checkpoints
Cell Differentiation
Cell Proliferation
Chondrosarcoma--metabolism
Enzyme Inhibitors--pharmacology
Glutarates--metabolism
Histone Code
Humans
Isocitrate Dehydrogenase--antagonists & inhibitors
Mutation
SOX9 Transcription Factor--metabolism