Kinetics of binding of membrane-active drugs to receptor sites. Diffusion-limited rates for a membrane bilayer approach of 1,4-dihydropyridine calcium channel antagonists to their active site.
Rhodes, D G
Kinetics of binding of membrane-active drugs to receptor sites. Diffusion-limited rates for a membrane bilayer approach of 1,4-dihydropyridine calcium channel antagonists to their active site. [electronic resource] - Molecular pharmacology Jun 1985 - 612-23 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
0026-895X
Animals
Calcium Channel Blockers--metabolism
Calcium Channels
Diffusion
Dihydropyridines
Kinetics
Ligands
Lipid Bilayers--metabolism
Mathematics
Models, Biological
Myocardium--metabolism
Pyridines--metabolism
Receptors, Nicotinic--metabolism
Sarcolemma--metabolism
Kinetics of binding of membrane-active drugs to receptor sites. Diffusion-limited rates for a membrane bilayer approach of 1,4-dihydropyridine calcium channel antagonists to their active site. [electronic resource] - Molecular pharmacology Jun 1985 - 612-23 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
0026-895X
Animals
Calcium Channel Blockers--metabolism
Calcium Channels
Diffusion
Dihydropyridines
Kinetics
Ligands
Lipid Bilayers--metabolism
Mathematics
Models, Biological
Myocardium--metabolism
Pyridines--metabolism
Receptors, Nicotinic--metabolism
Sarcolemma--metabolism