Discovery of velpatasvir (GS-5816): A potent pan-genotypic HCV NS5A inhibitor in the single-tablet regimens Vosevi

Link, John O

Discovery of velpatasvir (GS-5816): A potent pan-genotypic HCV NS5A inhibitor in the single-tablet regimens Vosevi [electronic resource] - Bioorganic & medicinal chemistry letters 08 2019 - 2415-2427 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2019.04.027 doi


Antiviral Agents--chemical synthesis
Carbamates--chemical synthesis
Dose-Response Relationship, Drug
Drug Combinations
Drug Discovery
Genotype
Hepacivirus--drug effects
Heterocyclic Compounds, 4 or More Rings--chemical synthesis
Humans
Macrocyclic Compounds--chemistry
Microbial Sensitivity Tests
Molecular Structure
Protease Inhibitors--chemical synthesis
Sofosbuvir--chemistry
Structure-Activity Relationship
Sulfonamides--chemistry
Tablets--chemistry
Viral Nonstructural Proteins--antagonists & inhibitors