Crystal structure of Plasmodium falciparum adenosine deaminase reveals a novel binding pocket for inosine.

Jaruwat, Aritsara

Crystal structure of Plasmodium falciparum adenosine deaminase reveals a novel binding pocket for inosine. [electronic resource] - Archives of biochemistry and biophysics 05 2019 - 6-13 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1096-0384

10.1016/j.abb.2019.04.002 doi


Adenosine Deaminase--chemistry
Adenosine Deaminase Inhibitors--chemistry
Amino Acid Sequence
Amino Acid Substitution
Catalytic Domain
Crystallography, X-Ray
Drug Design
Humans
Inosine--metabolism
Kinetics
Models, Molecular
Mutagenesis, Site-Directed
Plasmodium falciparum--enzymology
Protozoan Proteins--chemistry
Recombinant Proteins--chemistry
Sequence Homology, Amino Acid
Substrate Specificity