PROTAC-Mediated Degradation of Bruton's Tyrosine Kinase Is Inhibited by Covalent Binding.
Tinworth, Christopher P
PROTAC-Mediated Degradation of Bruton's Tyrosine Kinase Is Inhibited by Covalent Binding. [electronic resource] - ACS chemical biology 03 2019 - 342-347 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1554-8937
10.1021/acschembio.8b01094 doi
Adenine--analogs & derivatives
Agammaglobulinaemia Tyrosine Kinase--metabolism
Inhibitor of Apoptosis Proteins--metabolism
Piperidines
Protein Binding
Protein Kinase Inhibitors--chemistry
Proteolysis
Pyrazoles--chemistry
Pyrimidines--chemistry
Ubiquitin-Protein Ligases--metabolism
PROTAC-Mediated Degradation of Bruton's Tyrosine Kinase Is Inhibited by Covalent Binding. [electronic resource] - ACS chemical biology 03 2019 - 342-347 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1554-8937
10.1021/acschembio.8b01094 doi
Adenine--analogs & derivatives
Agammaglobulinaemia Tyrosine Kinase--metabolism
Inhibitor of Apoptosis Proteins--metabolism
Piperidines
Protein Binding
Protein Kinase Inhibitors--chemistry
Proteolysis
Pyrazoles--chemistry
Pyrimidines--chemistry
Ubiquitin-Protein Ligases--metabolism