Fluorine-18 isotope labeling for positron emission tomography imaging. Direct evidence for DBPR211 as a peripherally restricted CB1 inverse agonist.

Chang, Chun-Ping

Fluorine-18 isotope labeling for positron emission tomography imaging. Direct evidence for DBPR211 as a peripherally restricted CB1 inverse agonist. [electronic resource] - Bioorganic & medicinal chemistry 01 2019 - 216-223 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2018.11.043 doi


Animals
Cannabinoid Receptor Agonists--chemical synthesis
Drug Inverse Agonism
Fluorine Radioisotopes
Isotope Labeling
Male
Mice, Inbred C57BL
Positron-Emission Tomography--methods
Pyrazoles--chemical synthesis
Receptor, Cannabinoid, CB1--agonists
Sulfonamides--chemical synthesis
Thiophenes--chemistry
Tissue Distribution