Mode of binding of [3H]dibenzocycloalkenimine (MK-801) to the N-methyl-D-aspartate (NMDA) receptor and its therapeutic implication.

Kloog, Y

Mode of binding of [3H]dibenzocycloalkenimine (MK-801) to the N-methyl-D-aspartate (NMDA) receptor and its therapeutic implication. [electronic resource] - FEBS letters Mar 1988 - 167-70 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0014-5793

10.1016/0014-5793(88)80664-1 doi


2-Amino-5-phosphonovalerate
Animals
Anticonvulsants
Dibenzocycloheptenes--metabolism
Dizocilpine Maleate
Glutamates--pharmacology
Glutamic Acid
Glycine--pharmacology
Kinetics
Rats
Receptors, N-Methyl-D-Aspartate
Receptors, Neurotransmitter--drug effects
Valine--analogs & derivatives