Discovery of phenylalanine derivatives as potent HIV-1 capsid inhibitors from click chemistry-based compound library.

Wu, Gaochan

Discovery of phenylalanine derivatives as potent HIV-1 capsid inhibitors from click chemistry-based compound library. [electronic resource] - European journal of medicinal chemistry Oct 2018 - 478-492 p. digital

Publication Type: Journal Article

1768-3254

10.1016/j.ejmech.2018.09.029 doi


Anti-HIV Agents--chemical synthesis
Capsid--drug effects
Click Chemistry
HIV Infections--drug therapy
HIV-1--drug effects
Humans
Molecular Dynamics Simulation
Phenylalanine--analogs & derivatives
Small Molecule Libraries--chemical synthesis