Direct labelling of myocardial beta 1-adrenoceptors. Comparison of binding affinity of 3H-(-)-bisoprolol with its blocking potency.
Kaumann, A J
Direct labelling of myocardial beta 1-adrenoceptors. Comparison of binding affinity of 3H-(-)-bisoprolol with its blocking potency. [electronic resource] - Naunyn-Schmiedeberg's archives of pharmacology Oct 1985 - 27-39 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
0028-1298
10.1007/BF00498849 doi
Adenylyl Cyclases--metabolism
Adrenergic beta-Antagonists--metabolism
Animals
Binding, Competitive--drug effects
Bisoprolol
Catecholamines--pharmacology
Cats
Epinephrine--pharmacology
Female
Guinea Pigs
Heart Rate--drug effects
In Vitro Techniques
Male
Membranes--metabolism
Myocardial Contraction--drug effects
Myocardium--metabolism
Norepinephrine--pharmacology
Propanolamines--metabolism
Propranolol--pharmacology
Receptors, Adrenergic, beta--metabolism
Sinoatrial Node--drug effects
Stereoisomerism
Direct labelling of myocardial beta 1-adrenoceptors. Comparison of binding affinity of 3H-(-)-bisoprolol with its blocking potency. [electronic resource] - Naunyn-Schmiedeberg's archives of pharmacology Oct 1985 - 27-39 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
0028-1298
10.1007/BF00498849 doi
Adenylyl Cyclases--metabolism
Adrenergic beta-Antagonists--metabolism
Animals
Binding, Competitive--drug effects
Bisoprolol
Catecholamines--pharmacology
Cats
Epinephrine--pharmacology
Female
Guinea Pigs
Heart Rate--drug effects
In Vitro Techniques
Male
Membranes--metabolism
Myocardial Contraction--drug effects
Myocardium--metabolism
Norepinephrine--pharmacology
Propanolamines--metabolism
Propranolol--pharmacology
Receptors, Adrenergic, beta--metabolism
Sinoatrial Node--drug effects
Stereoisomerism