Benzofuro[3,2-d]pyrimidines inspired from cercosporamide CaPkc1 inhibitor: Synthesis and evaluation of fluconazole susceptibility restoration.
Dao, Viet Hung
Benzofuro[3,2-d]pyrimidines inspired from cercosporamide CaPkc1 inhibitor: Synthesis and evaluation of fluconazole susceptibility restoration. [electronic resource] - Bioorganic & medicinal chemistry letters 07 2018 - 2250-2255 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2018.05.044 doi
Antifungal Agents--chemical synthesis
Ascomycota--chemistry
Benzofurans--chemical synthesis
Biofilms--drug effects
Candida albicans--drug effects
Drug Resistance, Fungal--drug effects
Drug Synergism
Fluconazole--chemical synthesis
HeLa Cells
Humans
Protein Kinase C--antagonists & inhibitors
Protein Kinase Inhibitors--chemical synthesis
Pyrimidinones--chemical synthesis
Benzofuro[3,2-d]pyrimidines inspired from cercosporamide CaPkc1 inhibitor: Synthesis and evaluation of fluconazole susceptibility restoration. [electronic resource] - Bioorganic & medicinal chemistry letters 07 2018 - 2250-2255 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2018.05.044 doi
Antifungal Agents--chemical synthesis
Ascomycota--chemistry
Benzofurans--chemical synthesis
Biofilms--drug effects
Candida albicans--drug effects
Drug Resistance, Fungal--drug effects
Drug Synergism
Fluconazole--chemical synthesis
HeLa Cells
Humans
Protein Kinase C--antagonists & inhibitors
Protein Kinase Inhibitors--chemical synthesis
Pyrimidinones--chemical synthesis