Disposition of Mianserin and Cyclizine in UGT2B10-Overexpressing Human Embryonic Kidney 293 Cells: Identification of UGT2B10 as a Novel N-Glucosidation Enzyme and Breast Cancer Resistance Protein as an N-Glucoside Transporter.

Lu, Danyi

Disposition of Mianserin and Cyclizine in UGT2B10-Overexpressing Human Embryonic Kidney 293 Cells: Identification of UGT2B10 as a Novel N-Glucosidation Enzyme and Breast Cancer Resistance Protein as an N-Glucoside Transporter. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals 07 2018 - 970-979 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1521-009X

10.1124/dmd.118.080804 doi


ATP Binding Cassette Transporter, Subfamily G, Member 2--metabolism
Biological Transport--physiology
Cell Line
Cyclizine--metabolism
Glucosides--metabolism
Glucuronides--metabolism
Glucuronosyltransferase--metabolism
HEK293 Cells
Humans
Kidney--metabolism
Mianserin--metabolism
Multidrug Resistance-Associated Proteins--metabolism
Neoplasm Proteins--metabolism
RNA, Small Interfering--metabolism