Small molecule KDM4s inhibitors as anti-cancer agents.

Lin, Hongzhi

Small molecule KDM4s inhibitors as anti-cancer agents. [electronic resource] - Journal of enzyme inhibition and medicinal chemistry Dec 2018 - 777-793 p. digital

Publication Type: Journal Article

1475-6374

10.1080/14756366.2018.1455676 doi


Animals
Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
Enzyme Inhibitors--chemical synthesis
Humans
Jumonji Domain-Containing Histone Demethylases--antagonists & inhibitors
Lipopolysaccharides--antagonists & inhibitors
Macrophages--drug effects
Mice
Molecular Structure
RAW 264.7 Cells
Small Molecule Libraries--chemical synthesis
Structure-Activity Relationship
Tumor Necrosis Factor-alpha--antagonists & inhibitors