Sulfoximines as potent RORγ inverse agonists.

Ouvry, Gilles

Sulfoximines as potent RORγ inverse agonists. [electronic resource] - Bioorganic & medicinal chemistry letters 05 2018 - 1269-1273 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2018.03.041 doi


Animals
Drug Inverse Agonism
Female
Humans
Imines--chemical synthesis
Ligands
Mice, Inbred BALB C
Molecular Structure
Nuclear Receptor Subfamily 1, Group F, Member 3--antagonists & inhibitors
Stereoisomerism
Structure-Activity Relationship
Sulfonamides--chemical synthesis
Sulfoxides--chemical synthesis