Therapeutic targeting of membrane-associated GRP78 in leukemia and lymphoma: preclinical efficacy in vitro and formal toxicity study of BMTP-78 in rodents and primates.

Staquicini, D I

Therapeutic targeting of membrane-associated GRP78 in leukemia and lymphoma: preclinical efficacy in vitro and formal toxicity study of BMTP-78 in rodents and primates. [electronic resource] - The pharmacogenomics journal 05 2018 - 436-443 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1473-1150

10.1038/tpj.2017.46 doi


Animals
Cell Line, Tumor
Cell Survival--drug effects
Drug Evaluation, Preclinical
Endoplasmic Reticulum Chaperone BiP
Heat-Shock Proteins--antagonists & inhibitors
Humans
Leukemia--drug therapy
Lymphoma--drug therapy
Macaca fascicularis
Macaca mulatta
Mice
Molecular Targeted Therapy
Peptidomimetics--administration & dosage
Primates
Rats
United States
United States Food and Drug Administration