Discovery of a novel 2,4-dimethylquinoline-6-carboxamide M

Long, Madeline F

Discovery of a novel 2,4-dimethylquinoline-6-carboxamide M [electronic resource] - Bioorganic & medicinal chemistry letters 11 2017 - 4999-5001 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2017.10.016 doi


Allosteric Regulation
Amides--chemical synthesis
Animals
Brain--metabolism
Drug Evaluation, Preclinical
Half-Life
Protein Binding
Pyridines--chemistry
Rats
Rats, Sprague-Dawley
Receptor, Muscarinic M4--chemistry
Structure-Activity Relationship