Highly potent and selective Na

Storer, R Ian

Highly potent and selective Na [electronic resource] - Bioorganic & medicinal chemistry letters 11 2017 - 4805-4811 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2017.09.056 doi


Animals
Binding Sites
Dogs
Half-Life
Hepatocytes--metabolism
Humans
Infusions, Intravenous
Inhibitory Concentration 50
Mice
Microsomes, Liver--metabolism
Molecular Docking Simulation
NAV1.7 Voltage-Gated Sodium Channel--chemistry
Pain--drug therapy
Piperidines--chemistry
Protein Binding
Protein Structure, Tertiary
Pyridines--chemistry
Rats
Structure-Activity Relationship
Sulfonamides--chemistry
Thiadiazoles
Voltage-Gated Sodium Channel Blockers--chemistry