Development of an Inhibitor Screening Assay for Mono-ADP-Ribosyl Hydrolyzing Macrodomains Using AlphaScreen Technology.
Haikarainen, Teemu
Development of an Inhibitor Screening Assay for Mono-ADP-Ribosyl Hydrolyzing Macrodomains Using AlphaScreen Technology. [electronic resource] - SLAS discovery : advancing life sciences R & D 03 2018 - 255-263 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
2472-5560
10.1177/2472555217737006 doi
ADP-Ribosylation--drug effects
Adenosine Diphosphate Ribose--metabolism
Biological Assay--methods
Enzyme Inhibitors--pharmacology
Glycoside Hydrolases--antagonists & inhibitors
Humans
Hydrolysis--drug effects
Protein Processing, Post-Translational--drug effects
Proteins--metabolism
Development of an Inhibitor Screening Assay for Mono-ADP-Ribosyl Hydrolyzing Macrodomains Using AlphaScreen Technology. [electronic resource] - SLAS discovery : advancing life sciences R & D 03 2018 - 255-263 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
2472-5560
10.1177/2472555217737006 doi
ADP-Ribosylation--drug effects
Adenosine Diphosphate Ribose--metabolism
Biological Assay--methods
Enzyme Inhibitors--pharmacology
Glycoside Hydrolases--antagonists & inhibitors
Humans
Hydrolysis--drug effects
Protein Processing, Post-Translational--drug effects
Proteins--metabolism