Selective inhibition of PfA-M1, over PfA-M17, by an amino-benzosuberone derivative blocks malaria parasites development in vitro and in vivo.

Bounaadja, Lotfi

Selective inhibition of PfA-M1, over PfA-M17, by an amino-benzosuberone derivative blocks malaria parasites development in vitro and in vivo. [electronic resource] - Malaria journal 09 2017 - 382 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1475-2875

10.1186/s12936-017-2032-4 doi


Aminopeptidases--antagonists & inhibitors
Anisoles--pharmacology
Antimalarials--pharmacology
Cycloheptanes--pharmacology
Plasmodium falciparum--drug effects
Protease Inhibitors--pharmacology
Protozoan Proteins--antagonists & inhibitors