XE991 and Linopirdine Are State-Dependent Inhibitors for Kv7/KCNQ Channels that Favor Activated Single Subunits.

Greene, Derek L

XE991 and Linopirdine Are State-Dependent Inhibitors for Kv7/KCNQ Channels that Favor Activated Single Subunits. [electronic resource] - The Journal of pharmacology and experimental therapeutics 07 2017 - 177-185 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1521-0103

10.1124/jpet.117.241679 doi


Animals
Anthracenes--pharmacology
CHO Cells
Carbamates--pharmacology
Cricetinae
Cricetulus
Indoles--pharmacology
KCNQ1 Potassium Channel--antagonists & inhibitors
KCNQ2 Potassium Channel--drug effects
Kinetics
Membrane Potentials--drug effects
Mutation
Patch-Clamp Techniques
Phenylenediamines--pharmacology
Potassium Channel Blockers--pharmacology
Protein Subunits--drug effects
Pyridines--pharmacology
Rats