Discovery and structure activity relationship of the first potent cryptosporidium FIKK kinase inhibitor.

Osman, Khan T

Discovery and structure activity relationship of the first potent cryptosporidium FIKK kinase inhibitor. [electronic resource] - Bioorganic & medicinal chemistry 03 2017 - 1672-1680 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2017.01.036 doi


Amino Acid Sequence
Cryptosporidium--enzymology
Drug Discovery
Humans
Protein Kinase Inhibitors--chemistry
Protein Kinases--chemistry
Sequence Homology, Amino Acid
Spectrum Analysis--methods
Structure-Activity Relationship