Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease.

Jeřábek, Jakub

Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease. [electronic resource] - European journal of medicinal chemistry Feb 2017 - 250-262 p. digital

Publication Type: Journal Article

1768-3254

10.1016/j.ejmech.2016.12.048 doi


Acetylcholinesterase--metabolism
Alzheimer Disease--drug therapy
Amyloid beta-Peptides--chemistry
Animals
Antioxidants--chemistry
Blood-Brain Barrier--metabolism
Butyrylcholinesterase--metabolism
Cholinesterase Inhibitors--chemistry
Drug Design
Humans
Ligands
Liver--drug effects
Molecular Targeted Therapy
Neuroprotective Agents--chemistry
Peptide Fragments--chemistry
Protein Aggregates--drug effects
Rats
Resveratrol
Stilbenes--chemistry
Tacrine--chemistry